CHLOMIPHENE CITRATE :
Clomiphene (clomiphene citrate) is an anti-estrogenic medical substance. The use of clomiphene aims to increase the sperm cell count of semen. The substance is usually administered in 50 milligram daily doses during 2 to 3 months. In bodybuilding, clomid is used by athletes on the course of anabolic steroids to eliminate the side effects associated with the partial conversion of steroids to estrogen (female sex hormone), and to stimulate the internal production of testosterone after a course of steroids (at PCT), which is suppressed when taking steroids.
– one of the most common pharmacological drugs in the first-aid kit of bodybuilders on steroids. In this article, let’s talk about what is clomid, how the infertility medicine for women got into bodybuilding, we will give instructions on how to use it on the course of steroids and after it (on PCT), and also compare that tamoxifen or clomid is better.
What Is Clomid (Clomiphene Citrate)? Its Purpose
Clomid (clomiphene citrate) is a powerful antiestrogen, very similar in its effect to Tamoxifen (tamoxifen citrate).
Clomid (clomiphene citrate) is a powerful antiestrogen
Clomid gained great popularity in the 1970s in medicine as a drug for infertility in women and today it is still one of its main uses.
In bodybuilding, clomid is used by athletes on the course of anabolic steroids to eliminate the side effects associated with the partial conversion of steroids to estrogen (female sex hormone), and to stimulate the internal production of testosterone after a course of steroids (at PCT), which is suppressed when taking steroids.
1. Clomid Application In Medicine For Infertility
When taking clomiphene citrate, the levels of gonadotropin hormones in the blood increase.
Clomid use to treat infertility
Gonadotropins are a series of hormones (follicle-stimulating, luteinizing), which play an important role in regulating the function of the sexual glands. Through these hormones, the levels of testosterone and estrogen in the blood are controlled, which are known to determine the development and function of male and female genital organs.
With an increase in the level of gonadotropins, an egg is released in the body of the woman (ovulation occurs) and that is why the chance to become pregnant increases.
Clomid has been used in medicine since the 1970s to treat infertility in women.
2. Using Of Clomid In Bodybuilding On The Course Of Steroids
Clomid possesses strong anti-estrogenic properties, which can be useful in medicine and bodybuilding for athletes using steroids.
The fact is that testosterone and some steroids, obtained from testosterone, are partially converted into estrogen.
Elevated levels of estrogen leads to the development of gynecomastia (growth of the female breast) and excessive fluid retention in the body – both undesirable effects in bodybuilding.
Excess fluid increases blood pressure and hides muscle relief. That is why for its removal from the hypodermic layers on the drying of body professional bodybuilders take diuretics.
What makes clomid: when taken on a course of steroids, it blocks the receptors of estrogen in the body, preventing its action. Therefore, it can be useful for fighting gynecomastia, since the female breast is growing under the influence of estrogen.
How Useful Is Clomid For Bodybuilding?
Clomid in Bodybuilding on the Course of Steroids
According to information from the official site, the creators of which sell sports pharmacology and apparently understand well how it works:
“For serious users of steroids (those taking steroids regularly and in high doses) clomid is not effective enough to protect against the side effects of steroids associated with estrogen. They will need to take aromatase inhibitors that suppress the synthesis of estrogen. They are the most effective means to combat gynecomastia and water retention when taking steroids.”
With regard to fluid retention in the body: clomid may interfere with it to some extent, but it is not very effective for this, since it does not decrease the level of estrogen in the blood, but only “cuts off” the estrogen receptors.
It must however be understood that in most cases, water retention in the body is more a matter of proper nutrition than pharmacology. Excess carbohydrates in the diet, for example, helps to retain fluid in the body, which is further enhanced by the presence of anabolic steroids in the system.
Taking clomid on a course of steroids helps to avoid side effects associated with increased levels of estrogen (gynecomastia), but is ineffective in controlling fluid retention in the body.
3. Using Clomid In Bodybuilding After A Course Of Steroids On PCT
Most often, clomid in bodybuilding is used by athletes after a course of steroids at PCT (from the English PCT – Post Cycle Therapy – therapy after the course of steroids).
To accelerate the recovery of the natural production of testosterone, which is almost completely suppressed during the intake of anabolics. The degree of suppression is significantly dependent on the type of steroids and dose.
That is why almost all steroid courses include exogenous testosterone, but they are not limited to one. This is done in order to protect against the effects of low testosterone.
After stopping the use of steroids, the natural synthesis of testosterone begins to gradually recover, but the complete recovery takes quite a long time: from several months to a year.
PCT was designed specifically to help with the pharmacology process to restore the natural production of testosterone.
The most popular courses of PCT generally include clomid and tamoxifen, as well as peptide hormone – chorionic gonadotropin. Tamoxifen is an analogue of clomid according to antiestrogenic properties.
What does clomid do: it stimulates the release of gonadotropins, which in turn stimulates the natural production of testosterone.
– What happens if you do not do PCT after the course and do not take clomid?
At a minimum, you will have to fight the symptoms of low testosterone for a long time.
It is important to bear in mind that with reduced testosterone, the level of the catabolic hormone cortisol increases, under the influence of which the fat mass is more easily recruited and the muscular mass actively begins to degenerate.
PCT is recommended in the event that steroids are stopped for more than 8 weeks. If the break between courses (bridge) is less than 8 weeks or during it small doses of exogenous testosterone are injected, as is customary for hardcore athletes, but PCT can be avoided.
Clomiphene citrate is taken after a course of steroids on PCT to accelerate the restoration of the natural level of testosterone.
4. How Effective Is Clomid For Restoring Testosterone? Scientific Research
Scientific studies confirm that clomiphene citrate is really effective in increasing testosterone levels.
Taking clomiphene for 2 weeks by men aged 18-55 led to an approximately 2-fold increase in testosterone levels in most of them, but in some participants after 2 weeks and a month there was a sharp paradoxical drop in testosterone for scientists.
Clomid for Restoring Testosterone
A study of 125 men with low testosterone (less than 400 ng / dl) and decreased sexual desire, which took clomid for 3 months, showed that testosterone levels increased approximately twofold (from 309 ng / dL to 642 ng / dl). There were no changes in the level of cholesterol in the blood, side effects were also not noted by any of the participants 11.
And here 12 scientists have studied the long-term effect of taking clomid by men with low testosterone levels. At the beginning, the average testosterone level was 228 ng / dl. After one year of use, 612 ng / dl, after two years of 562 ng / dl, after three years of 582 ng / dl. Density of bones has considerably increased. There were no side effects.
Clomid significantly improves sexual function in men with hypogonadism and erectile dysfunction. Scientific studies confirm the effectiveness of clomid in increasing the level of testosterone on average by 2 times both with short-term admission (within 2 weeks) and with prolonged (for several years).
5. Side Effects Of Clomid In Bodybuilding
Clomid is considered one of the most well tolerated anti-estrogen in sports pharmacology and does not lead to serious side effects in either men or women. This is confirmed by scientific studies.
However, some side effects are possible.
Women who take clomiphene citrate for the treatment of infertility note at least the presence of one of the following side effects: irritability, sudden mood jumps, depression, water retention in the body.
Other possible side effects:
hot flashes (sudden temperature increase);
unpleasant sensations in the chest;
problems with vision;
When using clomid, visual impairment in the form of turbidity and blurring is possible. This is stated on the same site of the sports pharmacology store. It is also recommended in this case “to stop using it and then the vision will recover … in most cases.” There are several cases when this did not happen, most likely because Clomid was taken for a very long time in very high doses.”
In rats injections of clomid during pregnancy lead to multiple reproductive system disorders in offspring and mothers.
There is a possibility that taking clomiphene can lead to a decrease in bone density.
– Does clomid cause cancer?
Scientific studies do not confirm the relationship between the use of clomiphene citrate and the risk of cancer (breast, uterus and other forms), including long-term admission. It should be understood that almost all available studies have been conducted on women taking clomiphene for infertility treatment. There are no studies of athletes who are fond of pharmacology.
Clomid is considered a relatively safe anti-estrogen in bodybuilding. With his admission, visual impairment and a decrease in bone density are possible. Prolonged use does not increase the risk of developing cancer.
For athletes on the course of steroids to protect against estrogenic side effects, it is recommended to take 50 mg per day of clomid throughout the course. If this does not help, then it is unlikely that higher doses will be effective.
What Is Better: Clomid Or Tamoxifen On The Course Of Steroids?
According to information from the same steroid.com “many athletes note the greater efficacy of tamoxifen to protect against gynecomastia in the course of steroids. But in some cases it will not be possible to do without aromatase inhibitors. “
How To Take Clomid After A Course Of Steroids On PCT
After the course of steroids on PCT, clomid is taken as follows:
Week 1-2: a dose of 100-150 mg per day;
Week 3-4: a dose of 50-100 mg per day;
Week 5-6: dose of 50 mg per day.
The total duration of reception of clomid on PCT is 4-6 weeks. In most cases, tamoxifen and chorionic gonadotropin will be more effective.In order to test the effectiveness of clomiphene citrate on the course of PCT, you can take a blood test and make sure that the testosterone level is restored.
Many athletes note the greater effectiveness of tamoxifen compared with clomid on the course of steroids and after it.